[3+3] Annulative Functionalization Approaches to Poly-Functionalized 8-Acylindolizines, 8-Enylindolizines, and Indolizine-Coumarin Hybrids
  • Jeong, Yerin
  • Kim, Sunmi
  • Lee, Sunhee
  • 구도희
  • Oh, Hyunjin
  • 외 1명
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초록

Synthetic efforts to expand the indolizine chemical space via an annulative functionalization strategy are described. Cs2CO3-promoted [3 + 3] annulations under mild reaction conditions enabled facile decoration of a number of functional groups at the pyridine moiety by way of a domino N-alkylation-intramolecular aldol condensation procedure to afford a wide range of novel indolizines such as 8-acylindolizines, 8-enylindolizines, and coumarin-indolizine hybrids.

제목
[3+3] Annulative Functionalization Approaches to Poly-Functionalized 8-Acylindolizines, 8-Enylindolizines, and Indolizine-Coumarin Hybrids
저자
Jeong, YerinKim, SunmiLee, Sunhee구도희Oh, HyunjinKim, Ikyon
DOI
10.1021/acs.joc.5c00905
발행일
2025-07
저널명
Journal of Organic Chemistry
90
29
페이지
10282 ~ 10315